Protein List

Your search: Assay in [Protease inhibition]

Found 79 entries.


ID Name Class Organism Assay Summary
1 kalata B1 Cyclotide Viola odorata
Oldenlandia affinis
Viola tricolor
Hybanthus enneaspermus
Viola baoshanensis
Viola yedoensis
Viola philippica
Viola sumatrana Miq		 Kalata B1 and B2 were found to have no trypsin or chymotrypsin inhibitory activity. [...]
3 MCoTI-II Squash trypsin inhibitor Momordica cochinchinensis Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
4 kalata B2 Cyclotide Viola odorata
Oldenlandia affinis		 Kalata B1 and B2 were found to have no trypsin or chymotrypsin inhibitory activity. [...]
81 SFTI-1 BBI-like trypsin inhibitor Helianthus annus
Helianthus exilis
Helianthus tuberosus
Helianthus porteri
Helianthus praecox subsp. praecox
Helianthus schweinitzii		 Matriptase inhibitory activity of SFTI-2 is 25-fold less potent than native, while SFTI-3 exhibits similar potency. [...]
12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
Bifunctional analogues of SFTI-1 found to have trypsin and chymotrypsin inhibitory activity. [...]
SFTI-1 immobilised on gold and interaction with trypsin investigated. [...]
SFTI-1, an acyclic permutant and a [CYS-Abu]-cyclic mutant shown to possess potent trypsin inhibitory activity. [...]
SFTI-1 was found to have nano-molar inhibitory effect against matriptase and trypsin. [...]
Both SFTI-1 and acyclic SFTI-1 are potent inhibitors of bovine beta trypsin [...]
82 N-SFTI-1-C BBI-like trypsin inhibitor Synthetic Disulfide bond is essenial for structure and function of acyclic SFTI-1. Seleno aSFTI-1 has 30% reduced inhibitory constant. [...]
SFTI-1 and analogues shown to inhibit Bovine beta-trypsin and Human leukocyte elastase [...]
Chymotrypsin and trypsin Ka values determined for SFTI-1 analogues. [...]
SFTI-1, an acyclic permutant and a [CYS-Abu]-cyclic mutant shown to possess potent trypsin inhibitory activity. [...]
Both SFTI-1 and acyclic SFTI-1 are potent inhibitors of bovine beta trypsin [...]
83 SFTI-1(6,5) BBI-like trypsin inhibitor Synthetic SFTI-1(6,5) shown to have trypsin inhibitory activity and is cyclised after incubation with trypsin. [...]
93 [ABA3,11]SFTI-1 BBI-like trypsin inhibitor Synthetic SFTI-1 analogues assayed for trypsin inhibitory activity. [...]
SFTI-1, an acyclic permutant and a [CYS-Abu]-cyclic mutant shown to possess potent trypsin inhibitory activity. [...]
95 BiKK BBI-like trypsin inhibitor Synthetic Bifunctional analogues of SFTI-1 found to have trypsin and chymotrypsin inhibitory activity. [...]
96 BiKF BBI-like trypsin inhibitor Synthetic Bifunctional analogues of SFTI-1 found to have trypsin and chymotrypsin inhibitory activity. [...]
97 [ABA3,11]SFTI-1[6,5] BBI-like trypsin inhibitor Synthetic SFTI-1 analogues assayed for trypsin inhibitory activity. [...]
98 [ABA3,11]SFTI-1[1,14] BBI-like trypsin inhibitor Synthetic SFTI-1 analogues assayed for trypsin inhibitory activity. [...]
99 [Nlys5]SFTI-1 BBI-like trypsin inhibitor Synthetic Chymotrypsin and trypsin Ka values determined for SFTI-1 analogues. [...]
100 [Nphe5]SFTI-1 BBI-like trypsin inhibitor Synthetic Chymotrypsin and trypsin Ka values determined for SFTI-1 analogues. [...]
101 PP-SFTI-2 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
102 PP-SFTI-3 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
103 PP-SFTI-4 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
104 PP-SFTI-5 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
105 PP-SFTI-6 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
106 PP-SFTI-7 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
107 PP-SFTI-8 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
108 PP-SFTI-9 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
109 PP-SFTI-10 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
110 PP-SFTI-11 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
111 PP-SFTI-12 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
112 PP-SFTI-13 BBI-like trypsin inhibitor Synthetic Ki calculated for a range of SFTI-1 analogues against trypsin and chymotrypsin. [...]
137 MCoTI-I Squash trypsin inhibitor Momordica cochinchinensis Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
191 OSFEI I BBI-like trypsin inhibitor Synthetic SFTI based variants shown to have activity against Porcine pancreatic elastase and Proteinase K [...]
192 OSFEI II BBI-like trypsin inhibitor Synthetic SFTI based variants shown to have activity against Porcine pancreatic elastase and Proteinase K [...]
193 OSFPKI I BBI-like trypsin inhibitor Synthetic SFTI based variants shown to have activity against Porcine pancreatic elastase and Proteinase K [...]
194 OSFPKI II BBI-like trypsin inhibitor Synthetic SFTI based variants shown to have activity against Porcine pancreatic elastase and Proteinase K [...]
195 OSFPKI III BBI-like trypsin inhibitor Synthetic SFTI based variants shown to have activity against Porcine pancreatic elastase and Proteinase K [...]
196 HEI-TOS BBI-like trypsin inhibitor Synthetic SFTI based variants shown to have activity against Porcine pancreatic elastase and Proteinase K [...]
198 [Val5]SFTI-1 BBI-like trypsin inhibitor Synthetic SFTI-1 and analogues shown to inhibit Bovine beta-trypsin and Human leukocyte elastase [...]
199 [Ser5]SFTI-1 BBI-like trypsin inhibitor Synthetic SFTI-1 and analogues shown to inhibit Bovine beta-trypsin and Human leukocyte elastase [...]
200 [(R,S)HmVal5]SFTI-1 BBI-like trypsin inhibitor Synthetic SFTI-1 and analogues shown to inhibit Bovine beta-trypsin and Human leukocyte elastase [...]
201 [(S)HmVal5]SFTI-1 BBI-like trypsin inhibitor Synthetic SFTI-1 and analogues shown to inhibit Bovine beta-trypsin and Human leukocyte elastase [...]
202 [(R)HmVal5]SFTI-1 BBI-like trypsin inhibitor Synthetic SFTI-1 and analogues shown to inhibit Bovine beta-trypsin and Human leukocyte elastase [...]
203 [HmSer5]SFTI-1 BBI-like trypsin inhibitor Synthetic SFTI-1 and analogues shown to inhibit Bovine beta-trypsin and Human leukocyte elastase [...]
204 [G1A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
205 [R2A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
206 [T4A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
207 [K5A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
208 [S6A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
209 [I7A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
210 [P8A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
211 [P9A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
212 [I10A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
213 [F12A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
214 [P13A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
215 [D14A]SFTI-1 BBI-like trypsin inhibitor Synthetic 12 SFTI alanine mutants were tested for inhibitory activity against bovine trypsin. K5A mutant shows the weakest activity. [...]
216 Seleno aSFTI-1 BBI-like trypsin inhibitor Synthetic Disulfide bond is essenial for structure and function of acyclic SFTI-1. Seleno aSFTI-1 has 30% reduced inhibitory constant. [...]
217 [Ser3,11]aSFTI-1 BBI-like trypsin inhibitor Synthetic Disulfide bond is essenial for structure and function of acyclic SFTI-1. Seleno aSFTI-1 has 30% reduced inhibitory constant. [...]
218 SFTI-2 BBI-like trypsin inhibitor Synthetic Matriptase inhibitory activity of SFTI-2 is 25-fold less potent than native, while SFTI-3 exhibits similar potency. [...]
219 SFTI-3 BBI-like trypsin inhibitor Synthetic Matriptase inhibitory activity of SFTI-2 is 25-fold less potent than native, while SFTI-3 exhibits similar potency. [...]
226 oMCoTI-II Squash trypsin inhibitor Synthetic Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
227 [A10]oMCoTI-II Squash trypsin inhibitor Synthetic Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
228 [A13]oMCoTI-II Squash trypsin inhibitor Synthetic Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
229 [A14]oMCoTI-II Squash trypsin inhibitor Synthetic Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
230 [R10]oMCoTI-II Squash trypsin inhibitor Synthetic Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
231 [R13]oMCoTI-II Squash trypsin inhibitor Synthetic Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
232 [R14]oMCoTI-II Squash trypsin inhibitor Synthetic Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
233 [AlaG10]oMCoTI-II Squash trypsin inhibitor Synthetic Open chain variants have reduced inhibitory activity against bovine trypsin compared to native cyclic proteins. [...]
341 MCoTI-II[K10R] Squash trypsin inhibitor Synthetic Synthetic MCoTI-I and MCoTI-II are both extremely potent trypsin inhibitors. [K10R] mutant has essentially wild-type activity against trypsin, whilst [K10F] and [K10Q] mutants are less active. [K10F] is the only mutant to show significant activity against chymotrypsin in this assay. [...]
342 MCoTI-II[K10Q] Squash trypsin inhibitor Synthetic Synthetic MCoTI-I and MCoTI-II are both extremely potent trypsin inhibitors. [K10R] mutant has essentially wild-type activity against trypsin, whilst [K10F] and [K10Q] mutants are less active. [K10F] is the only mutant to show significant activity against chymotrypsin in this assay. [...]
343 MCoTI-II[K10F] Squash trypsin inhibitor Synthetic Synthetic MCoTI-I and MCoTI-II are both extremely potent trypsin inhibitors. [K10R] mutant has essentially wild-type activity against trypsin, whilst [K10F] and [K10Q] mutants are less active. [K10F] is the only mutant to show significant activity against chymotrypsin in this assay. [...]
1876 alca 1 Cyclotide Allexis cauliflora alac 1 and alac 2 have micromolar inhibitory activity for human prolyl oligopeptidase (POP). [...]
1877 alca 2 Cyclotide Allexis cauliflora alac 1 and alac 2 have micromolar inhibitory activity for human prolyl oligopeptidase (POP). [...]
1878 MCoFx1 Squash trypsin inhibitor Synthetic Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1879 cMCoFx1 Squash trypsin inhibitor Synthetic Inhibitory activity of cMCoFx1 against a panel of serine proteases [...]
Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1880 MCoFx2 Squash trypsin inhibitor Synthetic Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1881 cMCoFx2 Squash trypsin inhibitor Synthetic Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1882 MCoFx3 Squash trypsin inhibitor Synthetic Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1883 cMCoFx3 Squash trypsin inhibitor Synthetic Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1884 MCoFx4 Squash trypsin inhibitor Synthetic Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1885 cMCoFx4 Squash trypsin inhibitor Synthetic Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1886 MCoFx5 Squash trypsin inhibitor Synthetic Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1887 cMCoFx5 Squash trypsin inhibitor Synthetic Human beta-coagulation factor XIIa (FXIIa) inhibitory activity (Ki) of chemically synthesized MCoTI-II and acyclic or cyclic MCoFx1-5 [...]
1888 cMCoTI-fxL1 Squash trypsin inhibitor Synthetic Inhibitory activity of cMCoTI-fxL1 against a panel of serine proteases [...]
1889 cMCoTI-fxL5 Squash trypsin inhibitor Synthetic Inhibitory activity of cMCoTI-fxL5 against a panel of serine proteases [...]